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抗腫瘤抗生素是由微生物產(chǎn)生的具有抗腫瘤活性的化學(xué)物質(zhì)。這種微生物產(chǎn)生的抗生素具��(dú)特的分子�(jié)�(gòu)、新穎的作用�(jī)�和高效的生物活�[1]。目�,抗腫瘤抗生素的研究已取得多方面�(jìn)�,并且多種抗腫瘤抗生素應(yīng)用于臨床,均收到了良好的療效。如放線菌素�鹽酸阿霉素�表柔比星和博來霉素等[2][3]。百靈威作為專業(yè)試劑供應(yīng)�,供�(yīng)抗腫瘤抗生素、抗腫瘤化合物等多種�(chǎn)��

�(chǎn)品列�

�(chǎn)品編�(hào) 英文名稱 中文名稱 CAS 作用靶點(diǎn)
338112 Actinomycin D, 98% 放線菌素 D, 98% 50-76-0 N/A
113424 Doxorubicin hydrochloride, 98% 鹽酸阿霉�, 98% 25316-40-9 DNA topoisomerase II抑制�
194237 Epirubicin hydrochloride, 98% 表柔比星鹽酸�, 98% 56390-09-1 DNA topoisomerase II抑制�
573584 Geldanamycin, 99% 格爾德霉�, 99% 30562-34-6 HSP90抑制�
135072 Mithramycin A 光輝霉素A 18378-89-7 Polymerase抑制�
948477 Rapamycin, 98% 雷帕霉素, 98% 53123-88-9 mTOR抑制�
282611 Wortmannin, 98% 渥曼青霉�, 98% 19545-26-7 PI3K抑制�
BIZ0413 Zeocin 博來霉素 11031-11-1 DNA Synthesis抑制�

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References

[1] Wang L, Cheng X, Huang C, et al. Rapamycin protects cardiomyocytes against anoxia/reoxygenation injury by inducing autophagy through the PI3k/Akt pathway[J]. Journal of Huazhong University of Science and Technology [Medical Sciences], 2015, 35(1): 10-15.

[2] Baluk P, Yao L C, Flores J, et al. Rapamycin Reverses Lymphatic Abnormalities In A Transgenic Mouse Model Of Pulmonary Lymphangiectasia[M]//B52. NEONATAL LUNG DISEASE: FROM BENCH TO BABIES. American Thoracic Society, 2016: A3866-A3866.

[3] Das D, Rameshbabu A P, Ghosh P, et al. Biocompatible nanogel derived from functionalized dextrin for targeted delivery of doxorubicin hydrochloride to MG 63 cancer cells[J]. Carbohydrate Polymers, 2017, 171: 27-38.

 

�(chǎn)品列�

 

�(chǎn)品編�(hào) 英文名稱 中文名稱 CAS 作用靶點(diǎn)
381488 Ara-G hydrate, 98% 阿糖鳥苷, 98% 38819-10-2 DNA/RNA Synthesis抑制�
274584 Carboplatin, 98% 碳鉑, 98% 41575-94-4 DNA/RNA Synthesis抑制�
258050 2-Chloro-2'-deoxyadenosine, 99% 2-�-2'-脫氧腺苷, 99% 4291-63-8 DNA/RNA Synthesis抑制�
275688 cis-Diamineplatinum(II) dichloride, 99% 順式-二氨二氯化鉑, 99% 15663-27-1 DNA/RNA Synthesis抑制�
180939 5-Fluorouracil, 99% 5-氟尿嘧啶, 99% 51-21-8 DNA/RNA Synthesis抑制�
271269 Gemcitabine hydrochloride, 99% 鹽酸吉西他濱, 99% 122111-03-9 DNA/RNA Synthesis抑制�
251696 Oxaliplatin, 95% 奧沙利鉑, 95% 61825-94-3 DNA/RNA Synthesis抑制�
996037 Afatinib, 98% 阿法替尼, 98% 850140-72-6 EGFR抑制�
341249 Erlotinib, 98% 埃羅替尼, 98% 183321-74-6 EGFR抑制�
831262 Lapatinib, 98% 拉帕替尼, 98% 231277-92-2 EGFR抑制�
795123 Lapatinib ditosylate, 98% 二甲苯磺酸拉帕替�, 98% 388082-77-7 EGFR抑制�
625238 Entinostat, 99% 恩替諾特, 99% 209783-80-2 HDAC抑制�
837002 Panobinostat, 98% 帕比司他, 98% 404950-80-7 HDAC抑制�
303595 Trichostatin A, 98% 曲古柳菌素A, 98% 58880-19-6 HDAC抑制�
1349106 Ruxolitinib phosphate salt, 99% 魯索利替尼磷酸鹽, 99% 1092939-17-7 JAK抑制�
1430418 Tofacitinib citrate, 99% 檸檬酸托法替�, 99% 540737-29-9 JAK抑制�
912849 Tofacitinib, 99% 托法替尼, 99% 477600-75-2 JAK抑制�
951485 Ruxolitinib, 99% 魯索替尼, 99% 941678-49-5 JAK抑制�
369172 6-Amino-3-methylpurine, 90% 6-氨基-3-甲基嘌呤, 90% 5142-23-4 PI3K抑制�
268623 Quercetin, 98% 槲皮�, 98% 117-39-5 PI3K抑制�
812864 Axitinib, 98% 阿西替尼, 98% 319460-85-0 VEGFR2抑制�
1239124 Ponatinib, 99% 帕納替尼, 99% 943319-70-8 VEGFR2抑制�
814262 Vandetanib, 99% 凡德他尼, 99% 443913-73-3 VEGFR2抑制�
1109982 Vatalanib dihydrochloride, 99% 瓦他拉尼堿二鹽酸�, 99% 212141-51-0 VEGFR2抑制�

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腫瘤研究化合�

蛋白酶體抑制� 核心生化試劑
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